SMA Research Platform

Evidence graph for Spinal Muscular Atrophy

Biology-first target discovery
Christian Fischer / Bryzant Labs
14,766Targets
453Trials
84Drugs
7Datasets
6,987Sources
64,683Claims
72,052Evidence
29,649Hypotheses
TARGETproteinHomo sapiens

PAK4p21-Activated Kinase 4

Description

Alternative LIMK2 activator, group II PAK. Direct phosphorylation of LIMK2 leading to CFL2 inactivation.

Linked hypotheses (20)

  • Off-target candidate: **4AP_ampyra** → PAK4 (iPTM=0.959)
    mechanismconf 96%
  • Off-target candidate: **4AP_ampyra** → PAK4 (iPTM=0.957)
    mechanismconf 96%
  • Off-target candidate: **4AP_ampyra** → PAK4 (iPTM=0.952)
    mechanismconf 95%
  • Off-target candidate: **riluzole** → PAK4 (iPTM=0.936)
    mechanismconf 94%
  • PAK4_chembl_1 binds LIMK2_aC (Boltz-2 iPTM=0.944)
    targetconf 94%
  • [Protein Interaction] PAK4 is implicated in SMA pathogenesis based on 18 converging claims
    targetconf 91%
  • [Protein Interaction] PAK4 is implicated in SMA pathogenesis based on 18 converging claims
    targetconf 91%
  • [Protein Interaction] PAK4 is implicated in SMA pathogenesis based on 18 converging claims
    targetconf 91%
  • [Protein Interaction] PAK4 is implicated in SMA pathogenesis based on 18 converging claims
    targetconf 91%
  • [Protein Interaction] PAK4 is implicated in SMA pathogenesis based on 18 converging claims
    targetconf 91%
  • [Protein Interaction] PAK4 is implicated in SMA pathogenesis based on 18 converging claims
    targetconf 91%
  • [Protein Interaction] PAK4 is implicated in SMA pathogenesis based on 18 converging claims
    targetconf 91%
  • [Protein Interaction] PAK4 is implicated in SMA pathogenesis based on 18 converging claims
    targetconf 91%
  • [Protein Interaction] PAK4 is implicated in SMA pathogenesis based on 18 converging claims
    targetconf 91%
  • Off-target candidate: **4AP_ampyra** → PAK4 (iPTM=0.911)
    mechanismconf 91%
  • [Protein Interaction] PAK4 is implicated in SMA pathogenesis based on 18 converging claims
    targetconf 91%
  • [Protein Interaction] PAK4 is implicated in SMA pathogenesis based on 18 converging claims
    targetconf 91%
  • [Protein Interaction] PAK4 is implicated in SMA pathogenesis based on 18 converging claims
    targetconf 91%
  • [Protein Interaction] PAK4 is implicated in SMA pathogenesis based on 18 converging claims
    targetconf 91%
  • [Protein Interaction] PAK4 is implicated in SMA pathogenesis based on 18 converging claims
    targetconf 91%

Top compound hits (0)

No ranked compounds yet for PAK4.

Linked claims (50)

TypePredicateConfSource
drug targetboltz2_offtarget_iptm96%
drug targetboltz2_offtarget_iptm96%
drug targetboltz2_offtarget_iptm96%
drug targetboltz2_offtarget_iptm96%
drug targetboltz2_offtarget_iptm95%
drug targetboltz2_offtarget_iptm95%
drug targetboltz2_offtarget_iptm94%
drug targetboltz2_offtarget_iptm94%
drug targetboltz2_offtarget_iptm91%
drug targetboltz2_offtarget_iptm91%
drug targetboltz2_offtarget_iptm91%
drug targetboltz2_offtarget_iptm91%
drug targetboltz2_offtarget_iptm90%
drug targetboltz2_offtarget_iptm90%
drug targetboltz2_offtarget_iptm87%
drug targetboltz2_offtarget_iptm87%
drug targetboltz2_offtarget_iptm86%
drug targetboltz2_offtarget_iptm86%
drug targetboltz2_offtarget_iptm85%
drug targetboltz2_offtarget_iptm85%

Showing 20 of 50.

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